The construction of various functionalized aromatic and heteroaromatics via annulation and C-H activation plays a vital role in advanced synthetic organic chemistry. These compounds have shown a lot of biological activities and widely used for the development of new drugs and functional materials. Owing to their importance and usefulness, we have been interested in the synthesis of aromatics and heteroaromatics utilizing new methodologies. In this presentation, we describe a facile and efficient construction of biologically interesting and diverse aromatics and heteroaromatics via annulation and C-H activation developed by our group (Scheme 1).1-10
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